Clinical TrialID 6132

Drug-Drug Interaction Study of Qualaquin and Midazolam

NCT00785486

Healthy

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Record Fields

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Clinical Trial Id
6132
Evidence Id
6132
Core Evidence Id
6132
Source Clinical Trial Id
6118
Herb2 Clinical Trial Id
HBCT006118
Nct Id
NCT00785486
Title
Drug-Drug Interaction Study of Qualaquin and Midazolam
Status
Completed
Phase
Phase 1
Study Result
Yes
Study Condition
Healthy
Study Type
Interventional
Study Design
Allocation: NON_RANDOMIZED|Intervention Model: SINGLE_GROUP|Masking: NONE|Primary Purpose: BASIC_SCIENCE
Intervention
DRUG: Midazolam Alone|DRUG: Qualaquin (quinine) alone steady state|DRUG: Midazolam and Qualaquin at steady state
Intervention Allocation
Non_Randomized
Intervention Model
Single_Group
Intervention Mask
Intervention Purpose
Basic_Science
Gender
All
Age
Adult
Enrollment
24
Outcome Measure
Maximum Serum Concentration (Cmax), Maximum serum concentration(Cmax), Day 1 (Midazolam Alone), Day 9 (Qualaquin (quinine) Alone), Day 10 Midazolam with Qualaquin (quinine)|Area Under the Concentration Time Curve From Zero to T (AUC 0-t) for Midazolam and 1-hydroxy Midazolam at Baseline and With Qualaquin (Quinine) at Steady State., Area under the concentration time curve(AUC 0-t) calculated by the linear trapezoidal method from time 0 to 24 hours, for Midazolam and 1-hydroxy-midazolam on day 1 (midazolam alone) and day 10 (midazolam with Qualaquin -(quinine) at steady state to determine if a significant drug interaction occurs between midazolam and quinine, Days 1 and 10 at 0.167, 0.25, 0.5, 0.75, 1, 1.25, 1.5, 2, 3, 4, 6, 7.917, 12, 15 and 24 hours|Area Under the Concentration Time Curve From Zero to Infinity (AUC Inf) for Midazolam and 1 Hydroxy Midazolam Before (Day 1) and After (Day 10) Qualaquin (Quinine)., AUC inf for Midazolam and hydroxy-midazolam on day 1 (midazolam alone) and day 10 (midazolam with steady state Qualaquin(quinine)- the sum of AUC0-t plus the ratio of the last measured plasma concentration to the elimination rate constant to determine whether a significant drug interaction occurs between midazolam and quinine, Days 1 and 10 at 0.167, 0.25, 0.5, 0.75, 1, 1.25, 1.5, 2, 3, 4, 6, 7.917, 12, 15 and 24 hours|The Area Under the the Concentration Time Curve From Zero to Tau (0-8hrs) for Qualaquin (Quinine) AUC Tau Before and After Midazolam, Qualaquin (quinine) - AUC tau alone at steady state (day 9) and in the presence of coadministered midazolam 2 mg (day 10) over the dosing interval (0 - 8 hours), as calculated by the linear trapezoidal method., Days 9 and 10 at 0, 0.5, 1, 1.5, 2, 2.5, 3, 3.5, 4, 5, 6, 7, and 7.917 hours
Sponsor Collaborator
Mutual Pharmaceutical Company, Inc.
Funded By
INDUSTRY
Location
MDS Pharma Services, Phoenix, Arizona, 85044, United States
Other Id
MPC-001-07-1001
Start Date
2007-03
Primary Completion Date
2007-03
Completion Date
2007-03
First Posted
2008-11-05
Results First Posted
2009-07-08
Last Update Posted
2012-08-31
Study Document
Study Url
https://clinicaltrials.gov/study/NCT00785486
Title Cn
Title En
Drug-Drug Interaction Study of Qualaquin and Midazolam
Bilingual Status
semi_complete